Telotristat Etiprate

Overview

Telotristat Etiprate is a small molecule active pharmaceutical ingredient (ChEMBL CHEMBL3348963).

Patent & exclusivity (US)

Per the FDA Orange Book (1 approved US product), the latest listed US patent on Telotristat Etiprate expires 28 Feb 2031. Generic API sourcing typically opens up once these lapse.

Chemical identity

IUPAC name

2-benzamidoacetic acid;ethyl (2S)-2-amino-3-[4-[2-amino-6-[(1R)-1-[4-chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]phenyl]propanoate

Canonical SMILES

CCOC(=O)[C@H](CC1=CC=C(C=C1)C2=CC(=NC(=N2)N)O[C@H](C3=C(C=C(C=C3)Cl)N4C=CC(=N4)C)C(F)(F)F)N.C1=CC=C(C=C1)C(=O)NCC(=O)O

InChIKey

XSFPZBUIBYMVEA-CELUQASASA-N