Sebetralstat

Overview

Sebetralstat is a small molecule active pharmaceutical ingredient (ChEMBL CHEMBL5095248).

Patent & exclusivity (US)

Per the FDA Orange Book (1 approved US product), the latest listed US patent on Sebetralstat expires 26 Jan 2039 and exclusivity 3 Jul 2032. Generic API sourcing typically opens up once these lapse.

Chemical identity

IUPAC name

N-[(3-fluoro-4-methoxy-2-pyridinyl)methyl]-3-(methoxymethyl)-1-[[4-[(2-oxo-1-pyridinyl)methyl]phenyl]methyl]pyrazole-4-carboxamide

Canonical SMILES

COCC1=NN(C=C1C(=O)NCC2=NC=CC(=C2F)OC)CC3=CC=C(C=C3)CN4C=CC=CC4=O

InChIKey

KGMPDQIYDKKXRD-UHFFFAOYSA-N