Gabapentin Enacarbil

Overview

Gabapentin Enacarbil is a small molecule active pharmaceutical ingredient (ChEMBL CHEMBL1628502).

API suppliers (4)

Suppliers of Gabapentin Enacarbil evidenced by a US FDA Type II Drug Master File or an EU Certificate of Suitability (CEP). Sources: FDA DMF list, EDQM certification database.

• ALIVUS LIFE SCIENCES LTDIndia1 active DMF GMP on record
• DASAMI LAB PRIVATE LTDIndia1 active DMF GMP on record
• APITORIA PHARMA PRIVATE LTDIndia1 active DMF GMP on record
• Zydus Lifesciences LimitedIndia1 active DMF GMP on record

Patent & exclusivity (US)

Per the FDA Orange Book (2 approved US products), the latest listed US patent on Gabapentin Enacarbil expires 10 Jun 2029. Generic API sourcing typically opens up once these lapse.

Chemical identity

IUPAC name

2-[1-[[1-(2-methylpropanoyloxy)ethoxycarbonylamino]methyl]cyclohexyl]acetic acid

Canonical SMILES

CC(C)C(=O)OC(C)OC(=O)NCC1(CCCCC1)CC(=O)O

InChIKey

TZDUHAJSIBHXDL-UHFFFAOYSA-N