Etrasimod Arginine

Overview

Etrasimod Arginine is a small molecule active pharmaceutical ingredient (ChEMBL CHEMBL3989933).

API suppliers (1)

Suppliers of Etrasimod Arginine backed by a verifiable FDA Type II Drug Master File. Source: FDA quarterly DMF list.

• Cipla USA, Inc.USA1 active DMF

Patent & exclusivity (US)

Per the FDA Orange Book (1 approved US product), the latest listed US patent on Etrasimod Arginine expires 21 Jun 2036 and exclusivity 12 Oct 2028. Generic API sourcing typically opens up once these lapse.

Chemical identity

IUPAC name

(2R)-2-amino-5-(diaminomethylideneamino)pentanoic acid;2-[(3R)-7-[[4-cyclopentyl-3-(trifluoromethyl)phenyl]methoxy]-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]acetic acid

Canonical SMILES

C1CCC(C1)C2=C(C=C(C=C2)COC3=CC4=C(C=C3)NC5=C4CC[C@@H]5CC(=O)O)C(F)(F)F.C(C[C@H](C(=O)O)N)CN=C(N)N

InChIKey

GVPVVOSNDUAUKM-YMQOIHNTSA-N