Bremelanotide

Overview

Bremelanotide is a protein active pharmaceutical ingredient (ChEMBL CHEMBL2070241).

API suppliers (1)

Suppliers of Bremelanotide backed by a verifiable FDA Type II Drug Master File. Source: FDA quarterly DMF list.

• SHANGHAI SINUOTIDES BIOPHARMACEUTICAL CO LTDChina1 active DMF

Patent & exclusivity (US)

Per the FDA Orange Book (1 approved US product), the latest listed US patent on Bremelanotide expires 29 Apr 2041. Generic API sourcing typically opens up once these lapse.

Chemical identity

IUPAC name

(3S,6S,9R,12S,15S,23S)-15-[[(2S)-2-acetamidohexanoyl]amino]-9-benzyl-6-[3-(diaminomethylideneamino)propyl]-12-(1H-imidazol-5-ylmethyl)-3-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18-hexazacyclotricosane-23-carboxylic acid

Canonical SMILES

CCCC[C@@H](C(=O)N[C@H]1CC(=O)NCCCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC2=CN=CN2)CC3=CC=CC=C3)CCCN=C(N)N)CC4=CNC5=CC=CC=C54)C(=O)O)NC(=O)C

InChIKey

FFHBJDQSGDNCIV-MFVUMRCOSA-N